Tapentadol 100 mg Tablet Use, Indication, Side Effects, Dosage, Mechanism of Action, Price, Contra-Indications, Drug Interactions...

TERRADOL 100 TABLETS 

Tapentadol is a medication used primarily for the management of moderate to severe pain.

Tapentadol is used for moderate to severe pain.

Use and Indications of Tapentadol 100 mg Tablet :

• Pain Management: It is used to relieve moderate to severe acute pain, such as pain following surgery or injury, and chronic pain conditions.

Mechanism of Action of Terradol 100 Tablet:

• Mu-opioid Receptor Agonism: Similar to traditional opioid pain relievers, tapentadol activates mu-opioid receptors in the central nervous system to reduce the perception of pain.
• Norepinephrine Reuptake Inhibition: Unlike traditional opioids, tapentadol also inhibits the reuptake of norepinephrine, which helps to enhance pain relief.
• Tapentadol decreases the perception of pain by blocking the transmission of pain signals to the brain.

Side Effects  of Tapentadol 100 mg Tablet :

Common side effects of tapentadol include:

• Nausea
• Vomiting
• Constipation
• Headache
• Dizziness
• Drowsiness

Serious side effects can include respiratory depression (especially at higher doses), serotonin syndrome (when used with other serotonergic drugs), and potentially fatal overdose.

Contraindications  of Terradol 100 Tablet:

• Patients with significant respiratory depression
• Patients with paralytic ileus (intestinal obstruction)
• Patients who are concurrently using or have recently used MAO inhibitors

Drug Interactions of Tapentadol 100 mg Tablet :

• Other CNS Depressants: Such as alcohol, benzodiazepines, and other opioids, which can increase the risk of respiratory depression.
• Serotonergic Drugs: Can lead to serotonin syndrome when combined with SSRIs, SNRIs, or MAO inhibitors.

Dosage:

• Initial Dose: The typical starting dose for immediate-release tablets is 50 mg every 4-6 hours as needed for pain.
• Maintenance Dose: Depending on the severity of pain and individual response, doses may be adjusted.The maximum daily dose is usually 600 mg.

Tapentadol is a potent opioid analgesic with dual mechanisms of action, providing effective pain relief for moderate to severe pain. However, it carries risks of side effects and potential for abuse, so it should be used with caution and under medical supervision.

Always consult with a healthcare provider for personalized advice regarding the use of tapentadol, including appropriate dosing, monitoring for side effects, and potential interactions with other medications.

For Use of registered medical practitioner or a hospital only

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